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PMID: 3134971 Published · ppublish English Journal Article

The action of prostanoid receptor agonists and antagonists on smooth muscle and platelets.

British journal of pharmacology ·Vol. 94 ·No. 2 ·1988-06-00 ·Pages 591-601

Eglen RM, Whiting RL

Abstract

1. Prostanoid receptors have been characterized in a range of guinea-pig and rat smooth muscle and platelets, according to the scheme of Coleman et al., (1985a), using agonists (prostaglandin D2 (PGD2), PGE1, PGE2, 16,16 dimethyl PGE2, PGF2 alpha, PGI2 and U46619) and putative selective antagonists (AH 6809 and SQ 29,548). 2. The ileum possesses EP1- and IP-receptors; the trachea, EP1-EP2- and TP-receptors; the oesophageal muscularis mucosa, EP1- and TP-receptors; the aorta and the portal vein TP-receptors. The rat colon possesses IP-, FP- and TP-receptors. 3. Guinea-pig platelets possess both IP and DP receptors mediating an inhibition of aggregation and TP receptors mediating proaggregation responses. No evidence was found for the presence of EP1-, EP2- or FP-receptors. 4. Misoprostol and fenprostalene were characterized using the above preparations. Misoprostol acts as a selective EP1-agonist, and has little or no DP, FP, IP and TP activity. In the trachea precontracted with carbachol no evidence of EP2-receptor stimulation was observed. Fenprostalene possesses FP and TP activity but no EP1, EP2, DP or IP activity.

MeSH Terms
Alprostadil/analogs & derivatives,pharmacology Animals Aorta/physiology Blood Platelets/physiology Colon/physiology Esophagus/physiology Guinea Pigs In Vitro Techniques Male Misoprostol Muscle, Smooth/drug effects Platelet Aggregation/drug effects Portal Vein/physiology Prostaglandins F, Synthetic/pharmacology Rats Rats, Inbred Strains Receptors, Prostaglandin/analysis,drug effects Trachea/physiology
Chemicals
Prostaglandins F, Synthetic Receptors, Prostaglandin Misoprostol Alprostadil fenprostalene
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Eglen R M
Institute of Pharmacology, Syntex Research, Palo Alto, CA 94303.
Whiting R L
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17 references, click to expand
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Article Info
Journal
British journal of pharmacology
Abbr.
Br J Pharmacol
ISSN
0007-1188
Published
1988-06-00
Pages
591-601
Language
English
Region
England
NLM ID
7502536
PMCID
PMC1854006
Subset
IM
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