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PMID: 1000135 Published · ppublish English Comparative Study Journal Article

A comparison of affinity constants for muscarine-sensitive acetylcholine receptors in guinea-pig atrial pacemaker cells at 29 degrees C and in ileum at 29 degrees C and 37 degrees C.

British journal of pharmacology ·Vol. 58 ·No. 4 ·1976-12-00 ·Pages 613-20

Barlow RB, Berry KJ, Glenton PA, Nilolaou NM, Soh KS

Abstract

1 The affinity of 17 compounds for muscarine-sensitive acetylcholine receptors in atrial pacemaker cells and ileum of the guinea-pig has been measured at 29 degrees C in Ringer-Locke solution. Measurements were also made at 37 degrees C with 7 of them. 2 Some of the compounds had much higher affinity for the receptors in the ileum than for those in the atria. For the most selective compound, 4-diphenylacetoxy-N-methylpiperidine methiodide, the difference was approximately 20-fold. The receptors in the atria are therefore different the structure from those in the ileum. 3 The effect of temperature on affinity are not the same for all the compounds, tested indicating different enthalpies and entropies of adsorption and accounting for some of the difficulty experienced in predicting the affinity of new compounds.

MeSH Terms
Acetylcholine/physiology Animals Guinea Pigs Heart/drug effects Ileum/drug effects In Vitro Techniques Muscarine/pharmacology Organ Specificity Receptors, Drug/drug effects Temperature Thermodynamics Time Factors
Chemicals
Receptors, Drug Muscarine Acetylcholine
Authors & Affiliations
5 authors, click to expand affiliations / ORCID
Barlow R B
Berry K J
Glenton P A
Nilolaou N M
Soh K S
References (12)
12 references, click to expand
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Article Info
Journal
British journal of pharmacology
Abbr.
Br J Pharmacol
ISSN
0007-1188
Published
1976-12-00
Pages
613-20
Language
English
Region
England
NLM ID
7502536
PMCID
PMC1667484
Subset
IM
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