Abstract
UK-38,006, 6 beta-iodopenicillanic acid, was shown to be a potent inhibitor of beta-lactamase enzymes. It potentiated the antibacterial action of ampicillin in vitro against beta-lactamase-producing strains of Staphylococcus aureus, Haemophilus influenzae, Bacteroides fragilis. Neisseria gonorrhoeae, and many Enterobacteriaceae. This ability to synergize with ampicillin was also demonstrated in vivo after oral administration of UK-38,006 to experimentally infected mice. UK-38,006 was also shown to synergize in vitro with other penicillins and cephalosporins against beta-lactamase-producing strains of Escherichia coli, Proteus mirabilis, and Klebsiella species.
MeSH Terms
Ampicillin/pharmacology
Animals
Anti-Bacterial Agents/pharmacology
Bacteria/drug effects
Drug Synergism
Female
Mice
Microbial Sensitivity Tests
Penicillanic Acid/pharmacology
Penicillin Resistance
beta-Lactamase Inhibitors
Chemicals
Anti-Bacterial Agents
beta-Lactamase Inhibitors
Ampicillin
Penicillanic Acid
6-iodopenicillanic acid
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Moore B A
Brammer K W
References (10)
10 references, click to expand
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