Abstract
The D-alanine carboxypeptidase of Bacillus subtilis is a particulate enzyme that is irreversibly inactivated by penicillins and cephalosporins. However, the lethal concentrations of these antibiotics are not the same as those that inhibit enzymatic activity in vitro. 6-Aminopenicillanic acid inactivates at least 95% of the enzyme at nonlethal concentrations. Conversely, cephalothin is lethal at concentrations that do not inactivate the enzyme. Experiments with intact, growing cells confirm the results obtained in vitro. Therefore, a killing site distinct from the carboxypeptidase must be postulated.
MeSH Terms
Alanine
Bacillus subtilis/enzymology
Carboxypeptidases/antagonists & inhibitors
Cephalosporins/pharmacology
Cephalothin/pharmacology
Cloxacillin/pharmacology
Factor Analysis, Statistical
Hydrogen-Ion Concentration
Microbial Sensitivity Tests
Mutation
Penicillanic Acid/pharmacology
Penicillins/pharmacology
Peptidoglycan/antagonists & inhibitors
Structure-Activity Relationship
Time Factors
Chemicals
Cephalosporins
Penicillins
Peptidoglycan
Penicillanic Acid
Carboxypeptidases
Cloxacillin
Alanine
Cephalothin
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Blumberg P M
Strominger J L
References (6)
6 references, click to expand
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