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PMID: 32430 Published · ppublish English Journal Article

[3H] Dihydroergonine binding to alpha-adrenergic receptors in human platelets.

Klinische Wochenschrift ·Vol. 56 Suppl 1 ·1978-00-00 ·Pages 139-45

Jakobs KH, Rauschek R

Abstract

暂无摘要

MeSH Terms
Adrenergic alpha-Agonists/pharmacology Adrenergic alpha-Antagonists/blood,metabolism Binding Sites Blood Platelets/metabolism Catecholamines/pharmacology Cell Membrane/metabolism Ergoloid Mesylates/blood,metabolism Humans Kinetics Receptors, Adrenergic/blood Receptors, Adrenergic, alpha/blood,metabolism
Chemicals
Adrenergic alpha-Agonists Adrenergic alpha-Antagonists Catecholamines Receptors, Adrenergic Receptors, Adrenergic, alpha Ergoloid Mesylates
Authors & Affiliations
2 authors, click to expand affiliations / ORCID
Jakobs K H
Rauschek R
References (25)
25 references, click to expand
  1. Studies on the effect of adrenergic blocking drugs on catecholamine-induced platelet aggregation and uptake of noradrenaline and 5-hydroxytryptamine.
    Acta Physiol Scand. 1969 Jan-Feb;75(1):129-38 PMID: 5785133
  2. Alpha-adrenergic receptors on human platelets.
    Life Sci. 1977 Nov 15;21(10):1429-38 PMID: 200810
  3. Dynamic interaction of prostaglandin and norepinephrine in the formation of adenosine 3',5'-monophosphate in human and rabbit platelets.
    Biochim Biophys Acta. 1971 Feb 28;261(2):444-56 PMID: 4335547
  4. alpha-Adrenergic receptors in rat parotid cells. I. Correlation of [3H]dihydroergocryptine binding and catecholamine-stimulated potassium efflux.
    J Biol Chem. 1977 Aug 10;252(15):5472-7 PMID: 195950
  5. Aggregation of blood platelets by adenosine diphosphate and its reversal.
    Nature. 1962 Jun 9;194:927-9 PMID: 13871375
  6. Characterization of alpha- and beta-adrenergic receptors linked to human platelet adenylate cyclase.
    Naunyn Schmiedebergs Arch Pharmacol. 1978 May;302(3):285-91 PMID: 26887
  7. Characterization of the human platelet alpha-adrenergic receptor. Correlation of [3H]dihydroergocryptine binding with aggregation and adenylate cyclase inhibition.
    J Clin Invest. 1978 May;61(5):1136-44 PMID: 207726
  8. A functional basis for classification of alpha-adrenergic receptors.
    Life Sci. 1977 Sep 1;21(5):595-606 PMID: 20542
  9. The role of cyclic AMP in platelet function.
    Ann N Y Acad Sci. 1971 Dec 30;185:477-87 PMID: 4330513
  10. Identification of alpha-adrenergic receptors in human platelets by [3H]dihydroergocryptine binding.
    J Clin Invest. 1978 Feb;61(2):395-402 PMID: 23392
  11. Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reaction.
    Biochem Pharmacol. 1973 Dec 1;22(23):3099-108 PMID: 4202581
  12. Effects of catecholamines on the formation of adenosine 3':5'-cyclic monophosphate in human blood platelets.
    Biochem J. 1971 Nov;125(1):377-9 PMID: 4333938
  13. Protein measurement with the Folin phenol reagent.
    J Biol Chem. 1951 Nov;193(1):265-75 PMID: 14907713
  14. Identification of alpha-adrenergic receptors in uterine smooth muscle membranes by [3H]dihydroergocryptine binding.
    J Biol Chem. 1976 Nov 25;251(22):6915-23 PMID: 825511
  15. Inhibition of platelet adenylate cyclase by epinephrine requires GTP.
    FEBS Lett. 1978 Jan 1;85(1):167-70 PMID: 620788
  16. Platelet aggregation. 3. An epinephrine induced decrease in cyclic AMP synthesis.
    Biochem Biophys Res Commun. 1970 Jun 5;39(5):783-9 PMID: 4316427
  17. Pharmacological properties of (3H) dihydroergokryptine binding sites associated with alpha noradrenergic receptors in rat brain membranes.
    Mol Pharmacol. 1978 Jan;14(1):38-49 PMID: 203845
  18. Cyclic 3',5'-adenosine monophosphate in human blood platelets.
    Nature. 1969 Nov 8;224(5219):609-10 PMID: 4310361
  19. Effects of adrenaline on human blood platelets.
    J Physiol. 1967 Nov;193(2):443-53 PMID: 6065889
  20. Synthetic alpha-adrenergic agonists are potent alpha-adrenergic blockers in human platelets.
    Nature. 1978 Aug 24;274(5673):819-20 PMID: 28484
  21. SOME EFFECTS OF ADRENALINE AND ANTI-ADRENALINE COMPOUNDS ON PLATELETS IN VITRO AND IN VIVO.
    Nature. 1963 Nov 23;200:763-4 PMID: 14087010
  22. A COMPARISON OF PLATELET AGGREGATION PRODUCED BY SEVEN COMPOUNDS AND A COMPARISON OF THEIR INHIBITORS.
    J Clin Pathol. 1964 May;17:275-81 PMID: 14159460
  23. Reduction of adenylate cyclase activity in lysates of human platelets by the alpha-adrenergic component of epinephrine.
    J Cyclic Nucleotide Res. 1976 Nov-Dec;2(6):381-92 PMID: 14175
  24. [3H]Dihydroergocryptine binding to alpha adrenergic receptors in canine aortic membranes.
    J Pharmacol Exp Ther. 1978 Mar;204(3):606-14 PMID: 24730
  25. Characterization with [3H] dihydroergocryptine of the alpha-adrenergic receptor of the hepatic plasma membrane. Comparison with the beta-adrenergic receptor in normal and adrenalectomized rats.
    J Biol Chem. 1978 Feb 25;253(4):1114-20 PMID: 203582
Article Info
Journal
Klinische Wochenschrift
Abbr.
Klin Wochenschr
ISSN
0023-2173
DOI
10.1007/BF01477465
Published
1978-00-00
Pages
139-45
Language
English
Region
Germany
NLM ID
2985205R
Subset
IM
External Links
PubMed source DOI: 10.1007/BF01477465
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