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PMID: 19487463 Published · ppublish English Journal Article Research Support, N.I.H., Extramural Research Support, Non-U.S. Gov't

Site-specific mTOR phosphorylation promotes mTORC1-mediated signaling and cell growth.

Molecular and cellular biology ·Vol. 29 ·No. 15 ·2009-08-00 ·Pages 4308-24

Acosta-Jaquez HA, Keller JA, Foster KG, Ekim B, Soliman GA, Feener EP, Ballif BA, Fingar DC

Abstract

The mammalian target of rapamycin (mTOR) complex 1 (mTORC1) functions as a rapamycin-sensitive environmental sensor that promotes cellular biosynthetic processes in response to growth factors and nutrients. While diverse physiological stimuli modulate mTORC1 signaling, the direct biochemical mechanisms underlying mTORC1 regulation remain poorly defined. Indeed, while three mTOR phosphorylation sites have been reported, a functional role for site-specific mTOR phosphorylation has not been demonstrated. Here we identify a new site of mTOR phosphorylation (S1261) by tandem mass spectrometry and demonstrate that insulin-phosphatidylinositol 3-kinase signaling promotes mTOR S1261 phosphorylation in both mTORC1 and mTORC2. Here we focus on mTORC1 and show that TSC/Rheb signaling promotes mTOR S1261 phosphorylation in an amino acid-dependent, rapamycin-insensitive, and autophosphorylation-independent manner. Our data reveal a functional role for mTOR S1261 phosphorylation in mTORC1 action, as S1261 phosphorylation promotes mTORC1-mediated substrate phosphorylation (e.g., p70 ribosomal protein S6 kinase 1 [S6K1] and eukaryotic initiation factor 4E binding protein 1) and cell growth to increased cell size. Moreover, Rheb-driven mTOR S2481 autophosphorylation and S6K1 phosphorylation require S1261 phosphorylation. These data provide the first evidence that site-specific mTOR phosphorylation regulates mTORC1 function and suggest a model whereby insulin-stimulated mTOR S1261 phosphorylation promotes mTORC1 autokinase activity, substrate phosphorylation, and cell growth.

MeSH Terms
3T3-L1 Cells Adaptor Proteins, Signal Transducing/metabolism Animals Antibiotics, Antineoplastic/pharmacology Binding Sites/genetics Cell Cycle Proteins Cell Line Cell Proliferation Electrophoresis, Polyacrylamide Gel Flow Cytometry Humans Immunoblotting Immunoprecipitation Insulin/pharmacology Mass Spectrometry Mechanistic Target of Rapamycin Complex 1 Mice Multiprotein Complexes Phosphatidylinositol 3-Kinases/metabolism Phosphoinositide-3 Kinase Inhibitors Phosphoproteins/metabolism Phosphorylation/drug effects Protein Kinases/genetics,metabolism Proteins Signal Transduction/drug effects,genetics,physiology Sirolimus/pharmacology TOR Serine-Threonine Kinases Transcription Factors/genetics,metabolism
Chemicals
Adaptor Proteins, Signal Transducing Antibiotics, Antineoplastic Cell Cycle Proteins EIF4EBP1 protein, human Insulin Multiprotein Complexes Phosphoinositide-3 Kinase Inhibitors Phosphoproteins Proteins Transcription Factors Protein Kinases MTOR protein, human mTOR protein, mouse Mechanistic Target of Rapamycin Complex 1 TOR Serine-Threonine Kinases Sirolimus
Authors & Affiliations
8 authors, click to expand affiliations / ORCID
Acosta-Jaquez Hugo A
Department of Cell and Developmental Biology, University of Michigan Medical School, 109 Zina Pitcher Place, Ann Arbor, MI 48109-2200, USA.
Keller Jennifer A
Foster Kathryn G
Ekim Bilgen
Soliman Ghada A
Feener Edward P
Ballif Bryan A
Fingar Diane C
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Article Info
Journal
Molecular and cellular biology
Abbr.
Mol Cell Biol
ISSN
1098-5549
Published
2009-08-00
Epub
2009-00-01
Pages
4308-24
Language
English
Region
United States
NLM ID
8109087
PMCID
PMC2715808
Subset
IM
Grants
NCRR NIH HHS · P20 RR16462 · United States
NIDDK NIH HHS · R01 DK078135 · United States
NIDDK NIH HHS · 5P60 DK 20572 · United States
NIDDK NIH HHS · R01 DK-078135 · United States
NIDDK NIH HHS · P60 DK020572 · United States
NCRR NIH HHS · P20 RR016462 · United States
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